Appearance of new acetylcholine receptors on the baby chick biventer cervicis and denervated rat diaphragm muscles after blockade with α‐bungarotoxin

Abstract
1. The recovery of contractile responses and appearance of new alpha-bungarotoxin-binding sites were studied in the baby chick biventer cervicis and the rat diaphragm muscles after saturating the existing acetylcholine (ACh) receptors (AChR) with alpha-bungarotoxin in vitro.2. Washout of alpha-bungarotoxin restored gradually the response to exogenous ACh attaining about 30% recovery in 3 hr either in the chick muscle or in the denervated rat diaphragm. No recovery was obtained, however, for the response to nerve stimulation.3. The recovery of ACh-response was abolished by decreasing the bath temperature to 9 degrees C during the washout of the toxin whereas the recovery was not reduced in the presence of cycloheximide.4. The half-life of [(3)H]acetyl alpha-bungarotoxin bound specifically on the existing AChRs, junctional and extrajunctional receptors combined, was 16 hr in the chick muscle. That on the extrajunctional AChR was estimated to be 8 hr.5. New toxin-binding sites were found to be incorporated on the membrane of extrajunctional site rapidly after treatment with alpha-bungarotoxin in the chick and the denervated rat muscles along the muscle fibres but not in the innervated rat diaphragm. Treatment with (+)-tubocurarine, ACh or decamethonium did not cause an appreciable increase of the toxin-binding sites.6. The appearance of new binding sites was progressive during 5 hr at a rate of 24 sites/mum(2).hr in the chick muscle and 42 sites/mum(2).hr in the rat diaphragm denervated for 7 days. The existing extrajunctional AChR were about 50/mum(2) and 192/mum(2), respectively.7. ACh effectively antagonized the binding of alpha-bungarotoxin with the new sites whereas (+)-tubocurarine was less effective than its effect on the existing AChR.8. The new toxin-binding sites appeared to have a reduced capacity to evoke ACh response.9. The incorporation of new binding sites was reduced by lowering of the temperature, treatment with dinitrophenol, high K(+), high Ca(2+) and by the stimulation of either nerve or muscle. Cycloheximide, ACh, decrease of [Na(+)](o) and increase of [Mg(2+)](o) were without effect.10. It is suggested that binding of the extrajunctional AChRs with alpha-bungarotoxin cause a change of membrane architecture and trigger the incorporation of cytoplasmic AChR-precursor or hidden AChR into the membrane.