A simple strategy for the synthesis of hydroxyethylene dipeptide isostere from D-glucose

This publication has 18 references indexed in Scilit:

• Peptidomimetics—Tailored Enzyme Inhibitors
  Angewandte Chemie International Edition in English, 1994
• STRUCTURE-BASED INHIBITORS OF HIV-1 PROTEASE
  Annual Review of Biochemistry, 1993
• Hydroxyethylene isostere inhibitors of human immunodeficiency virus-1 protease: structure-activity analysis using enzyme kinetics, x-ray crystallography, and infected T-cell assays
  Biochemistry, 1992
• Stereocontrolled synthesis of HIV-1 protease inhibitors with C2-axis of symmetry
  Tetrahedron Letters, 1991
• Stereoselective synthesis of N-Boc-O-benzyl-(4S,5S)-5-amino-4-hydroxy-6-phenylhexanoic acid, the hydroxyethylene isosteric moiety of potent HIV-1 protease inhibitor
  Tetrahedron Letters, 1991
• Chapter 15. HIV Protease Inhibitors
  Published by Elsevier ,1991
• Synthesis of renin inhibitors possessing hydroxyethylene isostere residue from 3,4,6-tri-O-acetyl-D-qlucal via lactone precursor
  Tetrahedron, 1991
• Bis(tert-butylsulfonyl)acetylene as a general synthetic equivalent of alkynes in diels-alder chemistry. II: reductive and alkylative desulfonylations of bicyclic 1-alkyl-2-(tert-butylsulfonyl)ethenes
  Tetrahedron Letters, 1991
• A Synthetic HIV-1 Protease Inhibitor with Antiviral Activity Arrests HIV-Like Particle Maturation
  Science, 1990
• Inhibition of HIV-1 protease in infected T-lymphocytes by synthetic peptide analogues
  Nature, 1990