Synthesis and pharmacology of irreversible affinity labels as potential cocaine antagonists: aryl 1,4-dialkylpiperazines related to GBR-12783
- 22 September 1992
- journal article
- Published by Elsevier in European Journal of Pharmacology
- Vol. 220 (2-3) , 173-180
- https://doi.org/10.1016/0014-2999(92)90745-p
Abstract
No abstract availableKeywords
This publication has 24 references indexed in Scilit:
- Cloning and Expression of a Cocaine-Sensitive Rat Dopamine TransporterScience, 1991
- Dopamine transport sites selectively labeled by a novel photoaffinity probe: 125I-DEEPJournal of Neuroscience, 1989
- Ionic Requirements for the Specific Binding of [3H]GBR 12783 to a Site Associated with the Dopamine Uptake CarrierJournal of Neurochemistry, 1988
- Metaphit, a receptor acylator, inactivates cocaine binding sites in striatum and antagonizes cocaine-induced locomotor stimulation in rodentsNeuropharmacology, 1986
- High-affinity [3H]GBR 12783 binding to a specific site associated with the neuronal dopamine uptake complex in the central nervous systemEuropean Journal of Pharmacology, 1986
- Acylating phencyclidines irreversibly enhance brain calcium antagonist bindingPharmacology Biochemistry and Behavior, 1986
- Probes for narcotic receptor mediated phenomena. 7. Synthesis and pharmacological properties of irreversible ligands specific for .mu. or .delta. opiate receptorsJournal of Medicinal Chemistry, 1984
- Sodium‐Sensitive Cocaine Binding to Rat Striatal Membrane: Possible Relationship to Dopamine Uptake SitesJournal of Neurochemistry, 1983
- Quantitative aspects of hormone-receptor interactions of high affinity: Effect of receptor concentration and measurement of dissociation constants of labeled and unlabeled hormonesBiochimica et Biophysica Acta (BBA) - Biomembranes, 1975
- Reductions with Sulfurated Borohydrides. VI. The Reduction of Nitro, Nitrile, Amide, and Nitroso GroupsCanadian Journal of Chemistry, 1971