Penetration of 5-fluorouracil and prodrugs across the intestine of the albino rabbit: Evidence for shift in absorption site from the upper to the lower region of the gastrointestinal tract by prodrugs
- 1 September 1990
- journal article
- research article
- Published by Elsevier in Journal of Controlled Release
- Vol. 14 (1) , 43-51
- https://doi.org/10.1016/0168-3659(90)90059-3
Abstract
No abstract availableKeywords
This publication has 28 references indexed in Scilit:
- Clinical Pharmacology of 5-FluorouracilClinical Pharmacokinetics, 1989
- Biologic Activity of 5′-Deoxy-5-fluorouridine by Rectal AdministrationPharmaceutical Research, 1989
- Prodrugs of 5-fluorouracil. VIII. Improved rectal and oral delivery of 5-fluorouracil via various prodrugs. Structure-rectal absorption relationshipsInternational Journal of Pharmaceutics, 1987
- Intestinal Absorption of 5-Fluorouracil and its Alkylcarbamoyl Derivatives in the Rat Small IntestineJournal of Pharmaceutical Sciences, 1986
- Prodrugs of 5-Fluorouracil V. 1-Alkoxycarbonyl Derivatives as Potential Prodrug Forms for Improved Rectal or Oral Delivery of 5-FluorouracilJournal of Pharmaceutical Sciences, 1986
- Intestinal absorption characteristics of 5-fluorouracil, ftorafur and 6-mercaptopurine in rats.CHEMICAL & PHARMACEUTICAL BULLETIN, 1986
- Prodrugs of 5-fluorouracil. IV. Hydrolysis kinetics, bioactivation and physicochemical properties of various N-acyloxymethyl derivatives of 5-fluorouracilInternational Journal of Pharmaceutics, 1985
- Prodrugs of 5-fluorouracil. III. Hydrolysis kinetics in aqueous solution and biological media, lipophilicity and solubility of various 1-carbamoyl derivatives of 5-fluorouracilInternational Journal of Pharmaceutics, 1985
- Prodrugs of 5-fluorouracil. I. Hydrolysis kinetics and physicochemical properties of various N-acyl derivatives of 5-fluorouracilInternational Journal of Pharmaceutics, 1984
- Fluorouracil Therapy in Patients With Carcinoma of the Large BowelClinical Pharmacokinetics, 1978