An Enantioselective Synthesis of Cyclopentyl-L-Aspartic Acid Amenable to Large Scale

Abstract
A new enantioselective synthesis of cyclopentyl-L-aspartic acid[(S)-αamino-1-(carboxy)cyclopentaneacetic acid] (1) and its N-Boc derivative 2 has been developed. This synthesis is amenable to kilogram scale preparation and avoids low temperature reactions and column chromatography.

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