Some novel nucleoside rearrangements effected by (diethylamino)sulphur trifluoride: synthesis and antiviral properties of some fluorine-containing 3′-azido-3′-deoxythymidine derivatives
- 30 June 1993
- journal article
- Published by Elsevier in Journal of Fluorine Chemistry
- Vol. 62 (2-3) , 145-160
- https://doi.org/10.1016/s0022-1139(00)80089-5
Abstract
No abstract availableKeywords
This publication has 19 references indexed in Scilit:
- Some intramolecular rearrangements when pentofuranoses are treated with diethylaminosulphur trifluoride (DAST)Journal of Fluorine Chemistry, 1993
- Synthesis of 5′-O-phosphonomethyl-2′,3′-didehydro-2′,3′-dideoxyuridine by use of P-methoxybenzyl as a N3-protecting group.Tetrahedron Letters, 1991
- 4'-5'-Unsaturated 5'-halogenated nucleosides. Mechanism-based and competitive inhibitors of S-adenosyl-L-homocysteine hydrolaseJournal of Medicinal Chemistry, 1991
- Diethylaminosulfur trifluoride (DAST) as a fluorinating agent of pyrimidine nucleosides having a 2',3'-vicinal diol system.CHEMICAL & PHARMACEUTICAL BULLETIN, 1990
- Synthesis and antiviral activity of several 2,5'-anhydro analogs of 3'-azido-3'-deoxythymidine (AZT), 3'-azido-2',3'-dideoxyuridine (AZU), 3'-azido-2',3'-dideoxy-5-halouridines, and 3'-deoxythymidine against human immunodeficiency virus (HIV-1) and Rauscher-Murine leukemia virus (R-MuLV)Journal of Medicinal Chemistry, 1989
- 4',5'-Unsaturated-5'-fluoro adenosine nucleosides: potent mechanism-based inhibitors of S-adenosyl-L-homocysteine hydrolaseJournal of the American Chemical Society, 1989
- Synthesis and characterization of a new fluorine-substituted nonionic dinucleoside phosphonate analog. P-Deoxy-P-(difluoromethyl)thymidylyl(3' .fwdarw. 5')thymidineThe Journal of Organic Chemistry, 1988
- Synthesis of O2'-Methyluridine, O2'-Methylcytidine, N4,O2'-Dimethylcytidine and N4,N4,O2'-Trimethylcytidine from a Common Intermediate.Acta Chemica Scandinavica, 1986
- Regioselective reductive ring-opening of 4-methoxybenzylidene acetals of hexopyranosides. Access to a novel protecting-group strategy. Part 1Journal of the Chemical Society, Perkin Transactions 1, 1984
- 5‐Amino‐5‐deoxyribose derivatives. Synthesis and use in the preparation of “Reversed” NucleosidesJournal of Heterocyclic Chemistry, 1966