Synthesis and biological evaluation of the binding of dopamine D2/D3 receptor agonist, (R,S)-5-hydroxy-2-(N-propyl-N-(5′-18F-fluoropentyl)aminotetralin (18F-5-OH-FPPAT) in rodents and nonhuman primates

This publication has 9 references indexed in Scilit:

• Specific Binding of [¹¹C]Raclopride and N-[³H]Propyl-Norapomorphine to Dopamine Receptors in Living Mouse Striatum: Occupancy by Endogenous Dopamine and Guanosine Triphosphate–Free G Protein
  Journal of Cerebral Blood Flow & Metabolism, 2002
• (−)-N-[11C]propyl-norapomorphine: a positron-labeled dopamine agonist for PET imaging of D2 receptors
  Nuclear Medicine and Biology, 2000
• In vitro and in vivo evaluation of the binding of the dopamine D2 receptor agonist11C-(R,S)-5-hydroxy-2-(di-n-propylamino)tetralin in rodents and nonhuman primate
  Synapse, 2000
• Radiosynthesis and in vitro evaluation of 2-(N-alkyl-N-1′-11C-propyl)amino-5-hydroxytetralin analogs as high affinity agonists for dopamine D-2 receptors
  Nuclear Medicine and Biology, 1999
• Characterization of [I]S(−)5- binding to dopamine D2-like receptors expressed in cell lines
  Neuropharmacology, 1997
• Dopamine D2 receptors mapped in rat brain with [³H](+)PHNO
  Synapse, 1994
• Synthesis and in vivo distribution in the rat of several fluorine-18 labeled 5-hydroxy-2-aminotetralin derivatives
  Applied Radiation and Isotopes, 1993
• (R)‐ and (S)‐5‐hydroxy‐2‐(dipropylamino)tetralin (5‐OH DPAT): Assessment of optical purities and dopaminergic activities
  Chirality, 1990
• Complete Conversion of Brain D₂ Dopamine Receptors from the High‐ to the Low‐Affinity State for Dopamine Agonists, Using Sodium Ions and Guanine Nucleotide
  Journal of Neurochemistry, 1985