Design, synthesis and biological evaluation of pyridine-phenylpiperazines: A novel series of potent and selective α1a-adrenergic receptor antagonist

This publication has 42 references indexed in Scilit:

• The two-state model of receptor activation
  Trends in Pharmacological Sciences, 1995
• Modeling of G-protein-coupled receptors: application to dopamine, adrenaline, serotonin, acetylcholine, and mammalian opsin receptors
  Journal of Medicinal Chemistry, 1992
• Structural subtypes of the dopamine D2 receptor are functionally distinct: expression of the cloned D2A and D2B subtypes in a heterologous cell line
  Molecular Endocrinology, 1992
• Molecular biology of dopamine receptors
  Trends in Pharmacological Sciences, 1992
• Heterogeneity of [3H]-mepyramine binding sites in guinea pig cerebellum and lung
  Inflammation Research, 1991
• The efficacy and safety of terazosin for the treatment of symptomatic BPH
  The Prostate, 1991
• Molecular cloning and characterization of a novel dopamine receptor (D3) as a target for neuroleptics
  Nature, 1990
• Cloning and expression of a rat D2 dopamine receptor cDNA
  Nature, 1988
• The binding of [3H]nitrendipine to receptors for calcium channel antagonists in the heart, cerebral cortex, and ileum of rats
  Life Sciences, 1982
• Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction
  Biochemical Pharmacology, 1973