Simple Synthesis of 1-(Azacycloalkyl)Indoles Using Exclusive Ortho α-Chloroacetylation of N-(Azacycloalkyl)Anilines
- 1 February 1988
- journal article
- Published by Taylor & Francis in Synthetic Communications
- Vol. 18 (3) , 265-273
- https://doi.org/10.1080/00397918808057833
Abstract
Use of 2-(azacycloalkyl)amino-α-chloroacetophenones (4) as starting material makes possible simple synthesis of 1-(azacycloalkyl)-indoles (2).Keywords
This publication has 3 references indexed in Scilit:
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- Aminohaloborane in organic synthesis. 2. Simple synthesis of indoles and 1-acyl-3-indolinones using specific ortho .alpha.-chloroacetylation of anilinesThe Journal of Organic Chemistry, 1979
- Notiz über die Alkylierung des IndolsEuropean Journal of Inorganic Chemistry, 1954