Asymmetric total synthesis of a new non-natural 1β-methoxycarbapenem

Abstract
The asymmetric total synthesis of the new non-natural 1β-methoxycarbapenem (1) has been achieved via highly diastereoselective alkylation at the C-4 position of 4-acetoxyazetidin-2-one (4) with the tin enolate of thiazolidinethione (3); the stereochemistry has been confirmed by an X-ray crystal structure determination of the derivative (13).

This publication has 0 references indexed in Scilit: