β-Carbolines as inverse agonistic benzodiazepine receptor ligands. 2. Synthesis and in vitro and in vivo binding of some new 6-amino- and 6-fluoro-β-carboline-3-carboxylates
- 31 December 1995
- journal article
- research article
- Published by Elsevier in European Journal of Medicinal Chemistry
- Vol. 30 (3) , 245-251
- https://doi.org/10.1016/0223-5234(96)88232-8
Abstract
No abstract availableKeywords
This publication has 19 references indexed in Scilit:
- Synthesis of substituted 7,12-dihydropyrido[3,2-b:5,4-b']diindoles: rigid planar benzodiazepine receptor ligands with inverse agonist/antagonist propertiesJournal of Medicinal Chemistry, 1990
- New tetracyclic compounds containing the β‐carboline moietyJournal of Heterocyclic Chemistry, 1990
- β‐Carbolines as agonistic or antagonistic benzodiazepine receptor ligands.1. Synthesis of some 5‐, 6‐ and 7‐amino derivatives of 3‐methoxycarbonyl‐β‐carboline (β‐CCM) and of 3‐ethoxycarbonyl‐β‐carboline (β‐CCE)Journal of Heterocyclic Chemistry, 1988
- Topics in Phosphorus ChemistryOrganometallics, 1984
- Interaction of Convulsive Ligands with Benzodiazepine ReceptorsScience, 1982
- Is the benzodiazepine receptor coupled to a chloride anion channel?Nature, 1979
- Photochemistry of diazonium salts. II. Synthesis of 2-fluoro-L-histidine and 2-fluorohistamine, and the halogen lability of 2-fluoroimidazolesJournal of the American Chemical Society, 1973
- Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reactionBiochemical Pharmacology, 1973
- Photochemistry of diazonium salts. I. Synthesis of 4-fluoroimidazoles, 4-fluorohistamine, and 4-fluorohistidineJournal of the American Chemical Society, 1973
- THE ATTRACTIONS OF PROTEINS FOR SMALL MOLECULES AND IONSAnnals of the New York Academy of Sciences, 1949