A two-state receptor model for the interaction between angiotensin II type 1 receptors and non-peptide antagonists
- 6 February 2001
- journal article
- Published by Elsevier in Biochemical Pharmacology
- Vol. 61 (3) , 277-284
- https://doi.org/10.1016/s0006-2952(00)00546-3
Abstract
No abstract availableKeywords
This publication has 25 references indexed in Scilit:
- Mechanistic Differences of Various AT 1 -Receptor Blockers in Isolated Vessels of Different OriginHypertension, 1999
- Insurmountable angiotensin AT1 receptor antagonists: the role of tight antagonist bindingEuropean Journal of Pharmacology, 1999
- Binding of the antagonist []candesartan to angiotensin II AT1 receptor-tranfected Chinese hamster ovary cellsEuropean Journal of Pharmacology, 1999
- Distinction between surmountable and insurmountable selective AT1receptor antagonists by use of CHO-K1 cells expressing human angiotensin II AT1receptorsBritish Journal of Pharmacology, 1999
- Non-peptide Angiotensin Agonist: FUNCTIONAL AND MOLECULAR INTERACTION WITH THE AT1 RECEPTORPublished by Elsevier ,1995
- Agonist-antagonist interactions at angiotensin receptors: application of a two-state receptor modelTrends in Pharmacological Sciences, 1994
- Inhibition of rabbit aortic angiotensin II (AII) receptor by CV-11974, a new nonpeptide AII antagonistBiochemical Pharmacology, 1993
- Pharmacological profile of GR117289 in vitro: a novel, potent and specific non‐peptide angiotensin AT1 receptor antagonistBritish Journal of Pharmacology, 1992
- Evidence that the apparent complexity of receptor antagonism by angiotensin II analogues is due to a reversible and syntopic actionBritish Journal of Pharmacology, 1992
- The serotonin‐S2 Receptor: A receptor‐transducer coupling model to explain insurmountable antagonist effectsDrug Development Research, 1986