Novel 4,5,6,7-tetrahydrobenzothiazole dopamine agonists display very low stereoselectivity in their interaction with dopamine receptors.
- 31 December 1991
- journal article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 1 (4) , 189-192
- https://doi.org/10.1016/s0960-894x(00)80249-8
Abstract
No abstract availableKeywords
This publication has 6 references indexed in Scilit:
- Dopamine autoreceptor agonists as potential antipsychotics. 2. (Aminoalkoxy)-4H-1-benzopyran-4-onesJournal of Medicinal Chemistry, 1991
- Dopamine autoreceptor agonists: resolution and pharmacological activity of 2,6-diaminotetrahydrobenzothiazole and an aminothiazole analog of apomorphineJournal of Medicinal Chemistry, 1987
- Calculated and actual changes in β-adrenoceptor number associated with increases in rat and guinea-pig cardiac sensitivityJournal of Pharmacy and Pharmacology, 1986
- Identification of Dopamine "D3'' and "D4'' Binding Sites, Labelled with [3H]2-Amino-6,7-Dihydroxy- 1,2,3,4- Tetrahydronaphthalene, as High Agonist Affinity States of the D1 and D2 Dopamine Receptors, RespectivelyJournal of Neurochemistry, 1986
- Dopamine D2 receptor dissociation constant for spiperone: Identical values using 3H-labeled agonist or 3H-labeled antagonistBiochemical Pharmacology, 1985
- Dopaminergic neurons—Alteration in the sensitivity of tyrosine hydroxylase to inhibition by endogenous dopamine after cessation of impulse flowBiochemical Pharmacology, 1976