A Prodrug Approach to Increasing the Oral Potency of a Phenolic Drug. 1. Synthesis, Characterization, and Stability of an O-(lmidomethyl) Derivative of 17β-estradiol

This publication has 9 references indexed in Scilit:

• Mechanism of hydrolysis of O-imidomethyl derivatives of phenols
  The Journal of Organic Chemistry, 1993
• Phenyl carbamates of amino acids as prodrug forms for protecting phenols against first-pass metabolism
  International Journal of Pharmaceutics, 1992
• Mechanism of hydrolysis of benzamidomethyl derivatives of phenols and its implications for prodrug design
  The Journal of Organic Chemistry, 1992
• Prodrugs for Improved Oral β-Estradiol Bioavailability
  Pharmaceutical Research, 1988
• Prodrugs for improved oral nalbuphine bioavailability: inter-species differences in the disposition of nalbuphine and its acetylsalicylate and anthranilate esters
  International Journal of Pharmaceutics, 1987
• The metabolism of estradiol; oral compared to intravenous administration
  The Journal of Steroid Biochemistry and Molecular Biology, 1985
• Pharmacokinetics of Morphine and Its Surrogates II: Methods of Separation of Stabilized Heroin and Its Metabolites from Hydrolyzing Biological Fluids and Applications to Protein Binding and Red Blood Cell Partition Studies
  Journal of Pharmaceutical Sciences, 1979
• Reactivity of Nucleophilic Reagents toward Esters
  Journal of the American Chemical Society, 1960
• Struktur, Eigenschaften und Umsetzungen des Anlagerungsproduktes von Formaldehyd an Benzoesäure‐o‐sulfonsäureimid
  Archiv der Pharmazie, 1959