Efficient Syntheses of 4-Iodopyridine and of 4-Pyridylboronic Acid Pinacol Ester
- 1 October 1996
- journal article
- research article
- Published by Taylor & Francis in Synthetic Communications
- Vol. 26 (19) , 3543-3547
- https://doi.org/10.1080/00397919608003763
Abstract
4-iodopyridine can be prepared in good yield by low temperature diazotation-Sandmeyer reaction of the corresponding amine, then efficiently converted to the air-stable pinacol ester of 4-pyridylboronic acid.Keywords
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