Protective Effects of Ketotifen on Guinea Pig Trachea

Abstract
Effects were studied of ketotifen (Ke), an effective antiallergic drug, on guinea pig trachea. Ke (10-6-5 .times. 10-5 M) inhibits contractions induced in this preparation by acetylcholine, prostaglandin F2.alpha., BaCl2, KCl and electrical stimulation. Results suggest protective effects of Ke in airways. Ke exerts also a neural inhibitory effect on postganglionic parasympathetic fibers of guinea pig trachea. These findings resemble the effects reported previously for disodium cromoglycate and might be relevant for antiasthmatic and antiallergic properties of Ke.