A formal synthesis of (+)-lactacystin
- 19 September 2005
- journal article
- research article
- Published by Royal Society of Chemistry (RSC) in Chemical Communications
- Vol. 37 (40) , 5106-5108
- https://doi.org/10.1039/b508300a
Abstract
A synthetic route to the neurotrophic agent (+)-lactacystin has been developed utilizing a base-promoted intramolecular alkylidenecarbene C–H insertion as the key transformation.Keywords
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