Muscarinic agonists as analgesics. Antinociceptive activity versus M1 activity: SAR of alkylthio-TZTP's and related 1,2,5-thiadiazole analogs
- 10 February 1995
- journal article
- Published by Elsevier in Life Sciences
- Vol. 56 (11-12) , 807-814
- https://doi.org/10.1016/0024-3205(95)00014-w
Abstract
No abstract availableKeywords
This publication has 14 references indexed in Scilit:
- Cholinomimetics and Alzheimer's diseaseBioorganic & Medicinal Chemistry Letters, 1992
- Novel functional M1 selective muscarinic agonists. Synthesis and structure-activity relationships of 3-(1,2,5-thiadiazolyl)-1,2,5,6-tetrahydro-1-methylpyridinesJournal of Medicinal Chemistry, 1992
- Central muscarinic analgesia is mediated by M1 receptorsEuropean Journal of Pharmacology, 1990
- Direct binding studies on ileal and cardiac muscarinic receptorsBritish Journal of Pharmacology, 1987
- Identification of a Family of Muscarinic Acetylcholine Receptor GenesScience, 1987
- Pharmacological profile of a novel class of muscarinic acetylcholine receptor agonistsEuropean Journal of Pharmacology, 1986
- Alzheimer's Disease: A Disorder of Cortical Cholinergic InnervationScience, 1983
- Muscarinic receptor subtypes: M1 and M2 biochemical and functional characterizationLife Sciences, 1982
- A comparison of the antinociceptive actions of cholinomimetic and morphine‐like drugsBritish Journal of Pharmacology, 1970
- Studies on the central antinociceptive action of cholinomimetic agentsInternational Journal of Neuropharmacology, 1969