A Convenient Synthesis of Dialkyl [[2-(Bromomethyl)aziridin-1-yl]methyl]phosphonates, New Heterocyclic β-Azaphosphonates

Abstract
Dialkyl [[2-(bromomethyl)aziridin-1-yl]methyl] phosphonates were prepared in good yield by a convenient procedure involving the reaction of 1,3,5-triallylhexahydro[1,3,5]triazine with dialkyl phosphites, subsequent bromination and final ring closure upon treatment with sodium borohydride in methanol.

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