Enantioselective Synthesis of α,α′-Disubstituted Piperidines via Ruthenium-Catalyzed Ring Rearrangement

Abstract
A new method for the enantioselective synthesis of α,α′-disubstituted piperidines is described. Easily available cyclopentenones 5a,b rearrange via Ru-catalyzed RCM-ROM to heterocycles. Compound 6a is converted to the indolizidine 13.

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