Diastereoselective Synthesis of theC 2-Symmetric 2,3-Diaminotetralin via Electrophilic Amination
- 1 January 1994
- journal article
- research article
- Published by Georg Thieme Verlag KG in Synthesis
- Vol. 1994 (10) , 1026-1028
- https://doi.org/10.1055/s-1994-25629
Abstract
Starting from the N,N-dibenzyl protected ß-amino acid 3 a synthesis of the C 2-symmetric racemic 2,3-diaminotetralin (4; 2,3- diamino-1,2,3,4-tetrahydronaphthalene) is reported. The key step of the procedure is a highly stereocontrolled electrophilic amination by dibenzyl azodicarboxylate.Keywords
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