Inhibition of human leukocyte elastase by functionalized N-aryl azetidin-2-ones: substituent effects at C-3 and benzylic positions
- 31 December 1995
- journal article
- Published by Elsevier in European Journal of Medicinal Chemistry
- Vol. 30 (3) , 199-208
- https://doi.org/10.1016/0223-5234(96)88226-2
Abstract
No abstract availableKeywords
This publication has 27 references indexed in Scilit:
- Synthetic Inhibitors of ElastaseMedicinal Research Reviews, 1994
- Chapter 20. Proteinases in InflammationPublished by Elsevier ,1993
- Inhibition of human leukocyte elastase. 4. Selection of a substituted cephalosporin (L-658,758) as a topical aerosolJournal of Medicinal Chemistry, 1992
- Acyloxybenzyl halides, inhibitors of elastasesBiochimica et Biophysica Acta (BBA) - Protein Structure and Molecular Enzymology, 1991
- Monocyclic β-lactam inhibitors of human leukocyte elastaseTetrahedron, 1990
- Synthetic inhibitors of human neutrophil elastaseTrends in Pharmacological Sciences, 1987
- Inhibitors of leukocyte elastase and leukocyte Cathepsin G. Agents for the treatment of emphysema and related ailmentsMedicinal Research Reviews, 1987
- Cephalosporin antibiotics can be modified to inhibit human leukocyte elastaseNature, 1986
- Reaction of serine proteases with substituted 3-alkoxy-4-chloroisocoumarins and 3-alkoxy-7-amino-4-chloroisocoumarins: new reactive mechanism-based inhibitorsBiochemistry, 1985
- Interactions of Granulocyte Proteases with Inhibitors in Rheumatoid ArthritisPublished by Springer Nature ,1984