N-butyl, N-methyl, 11-[3′,17′ β-(dihydroxy)-1′,3′,5′(10′)- estratrien-16′ α-yl]-9(R/S)-bromo undecanamide: synthesis and 17β-HSD inhibiting, estrogenic and antiestrogenic activities

This publication has 23 references indexed in Scilit:

• 16α-propyl derivatives of estradiol as inhibitors of 17β-hydroxysteroid dehydrogenase type 1
  Bioorganic & Medicinal Chemistry Letters, 1994
• 11β-Amidoalkyl estradiols, a new series of pure antiestrogens
  The Journal of Steroid Biochemistry and Molecular Biology, 1992
• Expression of human 17β-hydroxysteroid dehydrogenase in mammalian cells
  The Journal of Steroid Biochemistry and Molecular Biology, 1992
• Distribution of 17β-hydroxysteroid dehydrogenase gene expression and activity in rat and human tissues
  The Journal of Steroid Biochemistry and Molecular Biology, 1992
• Synthesis and biological activity of new halo-steroidal antiestrogens
  Journal of Medicinal Chemistry, 1991
• Therapeutic potential of pure antioestrogens in the treatment of breast cancer
  The Journal of Steroid Biochemistry and Molecular Biology, 1990
• Endocrine Pharmacology of Antiestrogens as Antitumor Agents*
  Endocrine Reviews, 1990
• Antiestrogenic properties of keoxifene,trans-4-hydroxytamoxifen, and ICI 164384, a new steroidal antiestrogen, in ZR-75-1 human breast cancer cells
  Breast Cancer Research and Treatment, 1989
• Novel steroidal pure antiestrogens
  Steroids, 1989
• Mechanisms of oestrogen antagonism by nonsteroidal antioestrogens
  Molecular and Cellular Endocrinology, 1982