Studies on 2-Aziridinecarboxylic Acid. III. Reaction of 1-Acyl-2-aziridinecarboxylic Acid Peptide with Amines
- 1 January 1980
- journal article
- Published by Oxford University Press (OUP) in Bulletin of the Chemical Society of Japan
- Vol. 53 (1) , 283-284
- https://doi.org/10.1246/bcsj.53.283
Abstract
The reaction of Z–Gly–Azy–Gly–OBzl with amines was studied. With primary amines, the 1-acyl group (Z–Gly) of the aziridine peptide mainly migrated to the reactant amine with cleaving of the amide bond between glycine and aziridine, whereas aniline and diethylamine gave diaminopropionic acid derivatives via the ring opening reaction.Keywords
This publication has 3 references indexed in Scilit:
- Studies on 2-Aziridinecarboxylic Acid, II. A Novel Synthesis of Threonine O-Peptide Derivatives via (2S,3S)-3-Methyl-2-aziridinecarboxylic AcidBulletin of the Chemical Society of Japan, 1979
- Peptidsynthesen über N‐Phosphorylaminosäure‐phosphorsäure‐anhydrideEuropean Journal of Inorganic Chemistry, 1961
- Hydrogen Bonding and Basicity of Cyclic Imines1,2Journal of the American Chemical Society, 1956