Lack of tolerance to the anticonvulsant effects of tiagabine following chronic (21 day) treatment
- 31 December 1994
- journal article
- Published by Elsevier in Epilepsy Research
- Vol. 19 (3) , 205-213
- https://doi.org/10.1016/0920-1211(94)90063-9
Abstract
No abstract availableKeywords
This publication has 17 references indexed in Scilit:
- Discriminative stimulus effects of presynaptic GABA agonists in pentobarbital-trained ratsPharmacology Biochemistry and Behavior, 1994
- The synthesis of novel GABA uptake inhibitors. 1. Elucidation of the structure-activity studies leading to the choice of (R)-1-[4,4-bis(3-methyl-2-thienyl)-3-butenyl]-3-piperidinecarboxylic acid (Tiagabine) as an anticonvulsant drug candidateJournal of Medicinal Chemistry, 1993
- Tolerance to the anticonvulsant effects of carbamazepine, diazepam, and sodium valproate in kindled ratsPharmacology Biochemistry and Behavior, 1992
- Characterization of tiagabine (NO-328), a new potent and selective GABA uptake inhibitorEuropean Journal of Pharmacology, 1991
- Tolerance to the cognitive impairing effects but not the anticonvulsant effects of NO-328, a selective GABA uptake inhibitorEuropean Journal of Pharmacology, 1990
- (R)‐N‐[4,4‐Bis(3‐Methyl‐2‐Thienyl)but‐3‐en‐1‐yl]Nipecotic Acid Binds with High Affinity to the Brain γ‐Aminobutyric Acid Uptake CarrierJournal of Neurochemistry, 1990
- Tolerance to the anticonvulsant effect of benzodiazepinesTrends in Pharmacological Sciences, 1988
- GABA synaptic mechanisms: Stereochemical and conformational requirementsMedicinal Research Reviews, 1988
- Benzodiazepine cross-tolerance in mice extends to sodium valproateEuropean Journal of Pharmacology, 1986
- Biochemical and Electrophysiological Characteristics of Mammalian Gaba ReceptorsPublished by Elsevier ,1983