Synthesis of Functionalized Oxazolines and Oxazoles with DAST and Deoxo-Fluor
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- 25 March 2000
- journal article
- letter
- Published by American Chemical Society (ACS) in Organic Letters
- Vol. 2 (8) , 1165-1168
- https://doi.org/10.1021/ol005777b
Abstract
A mild and highly efficient cyclization of β-hydroxy amides to oxazolines is described using DAST and Deoxo-Fluor reagents. A one-pot protocol for the synthesis of oxazoles from β-hydroxy amides is also presented.Keywords
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