Palladium-Catalyzed Arylation and Heteroarylation of Indolizines
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- 28 February 2004
- journal article
- research article
- Published by American Chemical Society (ACS) in Organic Letters
- Vol. 6 (7) , 1159-1162
- https://doi.org/10.1021/ol049866q
Abstract
A highly effective protocol for palladium-catalyzed selective arylation and heteroarylation of indolizines at C-3 has been developed. Mechanistic studies unambiguously support an electrophilic substitution pathway for this transformation.Keywords
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