Enantioselective total synthesis of Glyoxalase I inhibitor using asymmetric Diels-Alder reaction of a new chiral dienophile, ()S-3-(3-triflouromethylpyrid-2-ylsulfinyl)acrylate.
- 1 January 1986
- journal article
- Published by Elsevier in Tetrahedron Letters
- Vol. 27 (45) , 5509-5512
- https://doi.org/10.1016/s0040-4039(00)85252-1
Abstract
No abstract availableKeywords
This publication has 10 references indexed in Scilit:
- Optically active 2--tolylsulfinylacrylate a novel chiral dienophile which exhibits high reactivity and diastereoselectivityTetrahedron Letters, 1985
- Synthesis of a Glyoxalase I Inhibitor from Streptomyces griseosporeus NIIDAet OGASAWARAHelvetica Chimica Acta, 1985
- Highly diastereoselective Diels-Alder reaction of optically active ethyl 2-p-tolylsulfinylmethylenepropionate with cyclopentadieneTetrahedron Letters, 1984
- Mechanism of action of 2-crotonyloxymethyl-4,5,6-trihydroxycyclohex-2-enone, a SH inhibitory antitumor antibiotic, and its effect on drug-resistant neoplastic cells.The Journal of Antibiotics, 1982
- The penems, a new class of .beta.-lactam antibiotics. 4. Syntheses of racemic and enantiomeric penem carboxylic acidsJournal of the American Chemical Society, 1979
- Simple syntheses of dl-phyllostine, dl-epoxydon and dl-epiepoxydonTetrahedron Letters, 1976
- The structure of a glyoxalase I inhibitor and its chemical reactivity with SH-compounds.The Journal of Antibiotics, 1975
- A glyoxalase I inhibitor of a new structural type produced by Streptomyces.The Journal of Antibiotics, 1975
- .alpha.-Methoxy-.alpha.-trifluoromethylphenylacetic acid, a versatile reagent for the determination of enantiomeric composition of alcohols and aminesThe Journal of Organic Chemistry, 1969
- Absolute Configuration and Optical Rotatory Power of Sulfoxides and Sulfinate Esters1,2Journal of the American Chemical Society, 1965