A [3H]amine congener of 1,3‐dipropyl‐8‐phenylxanthine
Open Access
- 21 April 1986
- journal article
- research article
- Published by Wiley in FEBS Letters
- Vol. 199 (2) , 269-274
- https://doi.org/10.1016/0014-5793(86)80493-8
Abstract
A xanthine amine congener (XAC), an amine‐functionalized derivative of 1,3‐dipropyl‐8‐phenylxanthine, is an antagonist ligand for A2 adenosine receptors of human platelets. XAC inhibited 5'‐N‐ethylca...Keywords
This publication has 19 references indexed in Scilit:
- Evidence for an A2 adenosine receptor in guinea pig lungNaunyn-Schmiedebergs Archiv für experimentelle Pathologie und Pharmakologie, 1985
- Ra Adenosine receptors in human plateletsNaunyn-Schmiedebergs Archiv für experimentelle Pathologie und Pharmakologie, 1984
- Effects of several 5?-carboxamide derivatives of adenosine on adenosine receptors of human platelets and rat fat cellsNaunyn-Schmiedebergs Archiv für experimentelle Pathologie und Pharmakologie, 1984
- A rapid filtration assay for soluble receptors using polyethylenimine-treated filtersAnalytical Biochemistry, 1983
- Functional identification of adenylate cyclase-coupled adenosine receptors in rat brain microvesselsEuropean Journal of Pharmacology, 1982
- Adenosine receptors: targets for future drugsJournal of Medicinal Chemistry, 1982
- Adenosine receptor agonists: Binding and adenylate cyclase stimulation in rat liver plasma membranesNaunyn-Schmiedebergs Archiv für experimentelle Pathologie und Pharmakologie, 1982
- 5′‐N‐ETHYLCARBOXAMIDOADENOSINE: A POTENT INHIBITOR OF HUMAN PLATELET AGGREGATIONBritish Journal of Pharmacology, 1981
- Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reactionBiochemical Pharmacology, 1973