Identification and characterization of 3-substituted pyrazolyl esters as alternate substrates for cathepsin B: The confounding effects of DTT and cysteine in biological assays
- 1 September 2007
- journal article
- research article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 17 (17) , 4761-4766
- https://doi.org/10.1016/j.bmcl.2007.06.091
Abstract
No abstract availableKeywords
This publication has 22 references indexed in Scilit:
- New Water-Soluble Phosphines as Reductants of Peptide and Protein Disulfide Bonds: Reactivity and Membrane PermeabilityBiochemistry, 2004
- Mechanism of action of pyridazine analogues on protein tyrosine phosphatase 1B (PTP1B)Bioorganic & Medicinal Chemistry Letters, 2004
- 4-Substituted d-Glutamic Acid Analogues: The First Potent Inhibitors of Glutamate Racemase (MurI) Enzyme with Antibacterial ActivityJournal of Medicinal Chemistry, 2002
- THE LYSOSOMAL CYSTEINE PROTEASESAnnual Review of Biophysics, 1999
- Novel Synthesis of 5-Amino-1-arylsulfonyl-4-pyrazolin-3-ones as a New Class of N-Sulfonylated PyrazolesJournal of Chemical Research, 1999
- Specific and Reversible Inactivation of Protein Tyrosine Phosphatases by Hydrogen Peroxide: Evidence for a Sulfenic Acid Intermediate and Implications for Redox RegulationBiochemistry, 1998
- Cysteine Proteases and Their InhibitorsChemical Reviews, 1997
- Attack of zwitterionic ammonium thiolates on a distorted anilide as a model for the acylation of papain by amides. A simple demonstration of a bell-shaped pH/rate profileJournal of the American Chemical Society, 1992
- Equilibrium acidities in dimethyl sulfoxide solutionAccounts of Chemical Research, 1988
- Selective method for the preparation of isomeric N‐alkyl and N‐aryl‐3(5)‐amino‐5(3)‐hydroxy‐1H‐pyrazole‐1‐carboxamidesJournal of Heterocyclic Chemistry, 1988