An Improved Procedure forN-Formylation of Secondary Amines Using Chlorotrimethylsilane-Imidazole-N,N-Dimethylformamide

Abstract
An improved method for the N-formylation of secondary amines using chlorotrimethylsilane and imidazole in N,N-dimethylformamide is described. The reaction conditions are tolerant of ester functional groups, and an amine hydrochloride may be N-formylated using a slight modification of the procedure.

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