E-17α-(2-[125I]IODOVINYL)-19-NORTESTOSTERONE: THE SYNTHESIS OF A GAMMA-EMITTING LIGAND FOR THE PROGESTERONE RECEPTOR.
- 1 December 1985
- journal article
- research article
- Published by The Endocrine Society in Endocrinology
- Vol. 117 (6) , 2550-2552
- https://doi.org/10.1210/endo-117-6-2550
Abstract
We have synthesized a gamma-emitting steroid, E-17.alpha.-(2-[125I]iodovinyl)-19-nortestosterone (E-IVNT), which is a useful ligand for the sensitive and accurate assay of the progesterone receptor. The synthetic scheme is rapid and is performed with readily available materials. This compund, [125I]E-IVNT, is stable and binds with high affinity to the progesterone receptor.This publication has 8 references indexed in Scilit:
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