An expeditious asymmetric synthesis of allophenylnorstatine
- 1 March 1994
- journal article
- Published by Elsevier in Tetrahedron
- Vol. 50 (13) , 3975-3986
- https://doi.org/10.1016/s0040-4020(01)89672-1
Abstract
No abstract availableKeywords
This publication has 19 references indexed in Scilit:
- Asymmetric syntheses of β-phenylalanine, α-methyl-β-phenylalanines and derivativesJournal of the Chemical Society, Chemical Communications, 1993
- Asymmetric synthesis of homochiral syn- and anti-3-phenylisoserine derivatives: a practical strategy for the synthesis of the taxol C-13 side chainJournal of the Chemical Society, Perkin Transactions 1, 1993
- Asymmetric Synthesis of AllophenylnorstatineSynlett, 1993
- Asymmetric synthesis of sulfinimines: applications to the synthesis of nonracemic .beta.-amino acids and .alpha.-hydroxyl .beta.-amino acidsThe Journal of Organic Chemistry, 1992
- Kynostatin (KNI-227 and -272, highly potent anti-HIV agents: conformationally constrained tripeptide inhibitors of HIV protease containing allophenylnorstatine.CHEMICAL & PHARMACEUTICAL BULLETIN, 1992
- HIV protease: a novel chemotherapeutic target for AIDSJournal of Medicinal Chemistry, 1991
- KNI-102, a novel tripeptide HIV protease inhibitor containing allophenylnorstatine as a transition-state mimic.CHEMICAL & PHARMACEUTICAL BULLETIN, 1991
- Rational design and synthesis of a novel class of active site-targeted HIV protease inhibitors containing a hydroxymethylcarbonyl isostere. Use of phenylnorstatine or allophenylnorstatine as a transition-state mimic.CHEMICAL & PHARMACEUTICAL BULLETIN, 1991
- Orally potent human renin inhibitors derived from angiotensinogen transition state: design, synthesis, and mode of interactionJournal of Medicinal Chemistry, 1990
- Synthesis and structure-activity relations of bestatin analogs, inhibitors of aminopeptidase BJournal of Medicinal Chemistry, 1977