A versatile approach to 2,3-disubstituted indoles through the palladium-catalysed cyclization of o-alkynyltrifluoroacetanilides with vinyl triflates and aryl halides.
- 1 June 1992
- journal article
- Published by Elsevier in Tetrahedron Letters
- Vol. 33 (27) , 3915-3918
- https://doi.org/10.1016/s0040-4039(00)74818-0
Abstract
No abstract availableThis publication has 14 references indexed in Scilit:
- Synthesis of indoles via palladium-catalyzed heteroannulation of internal alkynesJournal of the American Chemical Society, 1991
- Condensed Heteroaromatic Ring Systems; XVII:1Palladium-Catalyzed Cyclization of β-(2-Halophenyl)amino Substituted α,β-Unsaturated Ketones and Esters to 2,3-Disubstituted IndolesSynthesis, 1990
- Palladium-catalyzed synthesis of 2-substituted indolesThe Journal of Organic Chemistry, 1989
- Palladium-catalysed coupling of aryl and vinyl triflates or halides with 2-ethynylaniline: An efficient route to functionalized 2-substituted indolesTetrahedron Letters, 1989
- Palladium-catalyzed Indole and Benzofuran Ring Formation Accompanying CarbonylationHETEROCYCLES, 1989
- Palladium catalyzed reaction of 2-alkynylanilines with allyl chlorides. Formation of 3-allylindolesTetrahedron Letters, 1988
- Palladium-catalyzed coupling of 2-bromoanilines with vinylstannanes. A regiocontrolled synthesis of substituted indolesThe Journal of Organic Chemistry, 1988
- Synthesis of Condensed Heteroaromatic Compounds Using Palladium-Catalyzed ReactionHETEROCYCLES, 1988
- Synthesis of nitrogen heterocycles via palladium-catalyzed intramolecular cyclizationTetrahedron Letters, 1987
- Ortho-alkylation of acetanilides using alkyl halides and palladium acetateJournal of the American Chemical Society, 1984