Use of identical assay conditions for cocaine analog binding and dopamine uptake to identify potential cocaine antagonists

This publication has 15 references indexed in Scilit:

• Synthesis and Pharmacology of Potential Cocaine Antagonists. 2. Structure−Activity Relationship Studies of Aromatic Ring-Substituted Methylphenidate Analogs
  Journal of Medicinal Chemistry, 1996
• Hyperlocomotion and indifference to cocaine and amphetamine in mice lacking the dopamine transporter
  Nature, 1996
• Chimeric dopamine-norepinephrine transporters delineate structural domains influencing selectivity for catecholamines and 1-methyl-4-phenylpyridinium.
  Proceedings of the National Academy of Sciences, 1994
• Methoxylation of cocaine reduces binding affinity and produces compounds of differential binding and dopamine uptake inhibitory activity: discovery of a weak cocaine "antagonist"
  Journal of Medicinal Chemistry, 1993
• Studies of the biogenic amine transporters. II. A brief study on the use of [3H]DA-uptake-inhibition to transporter-binding-inhibition ratios for the in vitro evaluation of putative cocaine antagonists
  Life Sciences, 1993
• Cocaine and dopamine differentially protect [3H]mazindol binding sites from alkylation by N-ethylmaleimide
  European Journal of Pharmacology: Molecular Pharmacology, 1992
• Dopamine transporter site-directed mutations differentially alter substrate transport and cocaine binding.
  Proceedings of the National Academy of Sciences, 1992
• A multisubstrate mechanism of striatal dopamine uptake and its inhibition by cocaine
  Biochemical Pharmacology, 1992
• Kinetics and Block of Dopamine Uptake in Synaptosomes from Rat Caudate Nucleus
  Journal of Neurochemistry, 1990
• LIGAND: A versatile computerized approach for characterization of ligand-binding systems
  Analytical Biochemistry, 1980