(E)-1-(Heterocyclyl or cyclohexyl)-2-[1,3,7-trisubstituted (xanthin-8-yl)] ethenes as A2a adenosine receptor antagonists
- 31 December 1996
- journal article
- research article
- Published by Elsevier in European Journal of Medicinal Chemistry
- Vol. 31 (1) , 59-63
- https://doi.org/10.1016/s0223-5234(96)80007-9
Abstract
No abstract availableKeywords
This publication has 21 references indexed in Scilit:
- Synthesis of new pyrazolo[4,3-e]1,2,4-triazolo[1,5-c] pyrimidine and 1,2,3-triazolo[4,5-e]1,2,4-triazolo[1,5-c] pyrimidine displaying potent and selective activity as A2a adenosine receptor antagonists.Bioorganic & Medicinal Chemistry Letters, 1994
- KF17837 ((E)-8-(3,4-dimethoxystyryl)-1,3-dipropyl-7-methylxanthine) a potent and selective adenosine A2 receptor antagonistEuropean Journal of Pharmacology: Molecular Pharmacology, 1994
- Structure-activity relationships of 8-cycloalkyl-1,3-dipropylxanthines as antagonists of adenosine receptorsJournal of Medicinal Chemistry, 1990
- Optimization of parameters for semiempirical methods II. ApplicationsJournal of Computational Chemistry, 1989
- 7-Alkyltheophyllin-8-carbaldehydeCollection of Czechoslovak Chemical Communications, 1987
- Permanganate ion oxidations. 17. Kinetics and mechanism of the oxidation of (E)-3-(2-thienyl)-2-propenoates and (E)-3-(3-thienyl)-2-propenoates in phosphate-buffered solutionsJournal of the American Chemical Society, 1986
- Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reactionBiochemical Pharmacology, 1973
- 6-Phenylthieno[2,3-b]pyridine from 2-Nitro-3-thenaldehydeJournal of the American Chemical Society, 1957
- The Synthesis of Some β-Aminoethyldiazines as Histamine AnalogsJournal of the American Chemical Society, 1950
- 239. Fused carbon rings. Part XII. A simple synthesis of derivatives of decalin from cyclohexanone, and observations on cyclo-hexanespirobutyrolactone and allied compoundsJournal of the Chemical Society, 1937