Synthesis and pKa evaluation of model phosphonamidic, phosphonamidothioic, and phosphonamidodithioic acids
- 1 April 1996
- journal article
- Published by Elsevier in Tetrahedron
- Vol. 52 (17) , 6117-6124
- https://doi.org/10.1016/0040-4020(96)00274-8
Abstract
No abstract availableKeywords
This publication has 28 references indexed in Scilit:
- Synthesis of novel N-phosphonoalkyl dipeptide inhibitors of human collagenaseJournal of Medicinal Chemistry, 1994
- Phosphorus-containing inhibitors of endothelin converting enzyme: effects of the electronic nature of phosphorus on inhibitor potencyJournal of Medicinal Chemistry, 1993
- Transition-state structural features for the association of metalloproteases with phosphorus-containing inhibitorsJournal of the American Chemical Society, 1992
- Conformationally restricted P1-P1' transition state analogues. Synthesis of 1(R), 3(R) [1(S), 2(S)] and 1(S), 3(S) [1(S), 2(S)] 3-[3-cyclohexyl-2-[(BOC)amino]-1-hydroxypropyl]-2,2-dimethylcyclo propane carboxylic acidsTetrahedron Letters, 1990
- Potent inhibition of pepsin and penicillopepsin by phosphorus-containing peptide analogsThe Journal of Organic Chemistry, 1990
- Hydroxyethylamine analogs of the p17/p24 substrate cleavage site are tight-binding inhibitors of HIV proteaseJournal of Medicinal Chemistry, 1990
- Sequence-Specific Peptide Cleavage Catalyzed by an AntibodyScience, 1989
- Induction of an Antibody That Catalyzes the Hydrolysis of an Amide BondScience, 1988
- Evaluation of Intrinsic Binding Energy from a Hydrogen Bonding Group in an Enzyme InhibitorScience, 1987
- A phosphonamidate dipeptide analog as an inhibitor of carboxypeptidase AJournal of the American Chemical Society, 1981