Design and Synthesis of γ‐Dipeptide Derivatives with Submicromolar Affinities for Human Somatostatin Receptors
- 17 February 2003
- journal article
- research article
- Published by Wiley in Angewandte Chemie International Edition in English
- Vol. 42 (7) , 776-778
- https://doi.org/10.1002/anie.200390205
Abstract
No abstract availableKeywords
This publication has 22 references indexed in Scilit:
- Linear, Peptidase-Resistantβ2/β3-Di- andα/β3-Tetrapeptide Derivatives with Nanomolar Affinities to a Human Somatostatin Receptor, Preliminary CommunicationHelvetica Chimica Acta, 2001
- Design, Synthesis, NMR-Solution and X-Ray Crystal Structure ofN-Acyl-γ-dipeptide Amides That Form aβII′-Type TurnHelvetica Chimica Acta, 2001
- Somatostatin analogsChemical Biology & Drug Design, 2001
- Peptide Folding Induces High and Selective Affinity of a Linear and Small β-Peptide to the Human Somatostatin Receptor 4Journal of Medicinal Chemistry, 2001
- Identification of a Potent Heterocyclic Ligand To Somatostatin Receptor Subtype 5 by the Synthesis and Screening of β-Turn Mimetic LibrariesJournal of the American Chemical Society, 1999
- Potent Antagonists of Somatostatin: Synthesis and BiologyJournal of Medicinal Chemistry, 1998
- γ‐Peptides Forming More Stable Secondary Structures than α‐Peptides: Synthesis and helical NMR‐solution structure of the γ‐hexapeptide analog of H‐(Val‐Ala‐Leu)2‐OHHelvetica Chimica Acta, 1998
- Classification and nomenclature of somatostatin receptorsTrends in Pharmacological Sciences, 1995
- Conformation of two somatostatin analogues in aqueous solutionEuropean Journal of Biochemistry, 1989
- Conformational modifications of cyclic hexapeptide somatostatin analogsInternational Journal of Peptide and Protein Research, 1984