Simple One-Flask Method for the Preparation of Hydroxamic Acids
- 1 July 2003
- journal article
- Published by American Chemical Society (ACS) in Organic Letters
- Vol. 5 (15) , 2715-2717
- https://doi.org/10.1021/ol034903j
Abstract
[reaction: see text] A one-step conversion of carboxylic acids to hydroxamic acids under very mild conditions is described. This simple and efficient method has been applied for the synthesis of enantiopure hydroxamate of alpha-amino acids and peptides.Keywords
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