Generation of a piperazine-2-carboxamide library: A practical application of the phenol-sulfide react and release linker
- 1 March 1998
- journal article
- Published by Elsevier in Tetrahedron Letters
- Vol. 39 (11) , 1295-1298
- https://doi.org/10.1016/s0040-4039(97)10870-x
Abstract
No abstract availableKeywords
This publication has 12 references indexed in Scilit:
- Nucleoside transport inhibition by draflazine in unstable coronary diseaseEuropean Journal of Clinical Pharmacology, 1996
- A 24-week open-label Phase I/II evaluation of the HIV protease inhibitor MK-639 (indinavir)AIDS, 1996
- Activation Method to Prepare a Highly Reactive Acylsulfonamide “Safety-Catch” Linker for Solid-Phase Synthesis1Journal of the American Chemical Society, 1996
- Asymmetric hydrogenation of tetrahydropyrazines: Synthesis of (S)-piperazine-2-tert-butylcarboxamide, an intermediate in the preparation of the HIV protease inhibitor indinavirTetrahedron Letters, 1995
- Carbon-Carbon Bond-Forming Methods on Solid Support. Utilization of Kenner's "Safety-Catch" LinkerJournal of the American Chemical Society, 1994
- A conventient solid phase preparation of peptide substituted amidesTetrahedron Letters, 1994
- Multicyclic polypeptide model compounds. 1. Synthesis of a tricyclic amphiphilic .alpha.-helical peptide using an oxime resin, segment-condensation approachJournal of the American Chemical Society, 1990
- Polymer-bound oxime esters as supports for solid-phase peptide synthesis. The preparation of protected peptide fragmentsThe Journal of Organic Chemistry, 1980
- The safety catch principle in solid phase peptide synthesisJournal of the Chemical Society D: Chemical Communications, 1971
- Modified support for solid-phase peptide synthesis which permits the synthesis of protected peptide fragmentsThe Journal of Organic Chemistry, 1970