Probing of the cis-5-phenyl proline scaffold as a platform for the synthesis of mechanism-based inhibitors of the Staphylococcus aureus sortase SrtA isoform
- 13 February 2009
- journal article
- Published by Elsevier in Bioorganic & Medicinal Chemistry
- Vol. 17 (7) , 2886-2893
- https://doi.org/10.1016/j.bmc.2009.02.008
Abstract
No abstract availableKeywords
This publication has 26 references indexed in Scilit:
- Identification of novel inhibitors of bacterial surface enzyme Staphylococcus aureus Sortase ABioorganic & Medicinal Chemistry Letters, 2008
- Activation of Inhibitors by Sortase Triggers Irreversible Modification of the Active SiteJournal of Biological Chemistry, 2007
- A generally applicable method for assessing the electrophilicity and reactivity of diverse nitrile-containing compoundsBioorganic & Medicinal Chemistry Letters, 2006
- Vinyl sulfones: Synthetic preparations and medicinal chemistry applicationsMedicinal Research Reviews, 2006
- Stereoselective synthesis of functional derivatives of 2-(2-carboxyethyl)pyrrolidine-2-carboxylic acidRussian Journal of Organic Chemistry, 2006
- Bad Bugs Need Drugs: An Update on the Development Pipeline from the Antimicrobial Availability Task Force of the Infectious Diseases Society of AmericaClinical Infectious Diseases, 2006
- Bis(indole) alkaloids as sortase A inhibitors from the sponge Spongosorites sp.Bioorganic & Medicinal Chemistry Letters, 2005
- A Short Synthesis of 1-Vinyluracil and 1-VinylthymineSynthetic Communications, 1997
- Phase annealing in SHELX-90: direct methods for larger structuresActa Crystallographica Section A Foundations of Crystallography, 1990
- Prototropic routes to 1,3- and 1,5-dipoles, and 1,2-ylides: applications to the synthesis of heterocyclic compoundsChemical Society Reviews, 1987