Aromatic and Amine Substituent Effects on the Apparent Lipophiiicities of N-[(2-Pyrrolidinyl)methyl]-Substituted Benzamides

This publication has 41 references indexed in Scilit:

• Fluorinated benzamide neuroleptics—2. Synthesis and radiosynthesis of (S)-N-[(1-ethyl-2-pyrrolidinyl)methyl]-5-(3-[18F]fluoropropyl)-3-substituted-2-methoxybenzamides
  International Journal of Radiation Applications and Instrumentation. Part A. Applied Radiation and Isotopes, 1991
• High affinity dopamine D2 receptor radioligands. 2. [125I]epidepride, a potent and specific radioligand for the characterization of striatal and extrastriatal dopamine D2 receptors
  Life Sciences, 1991
• Preparation of [¹²³I]‐ and [¹²⁵I]epidepride: A dopamine D‐2 receptor antagonist radioligand
  Journal of Labelled Compounds and Radiopharmaceuticals, 1991
• Fluorinated benzamide neuroleptics. 1. Radiosynthesis of (S)‐N‐[(1‐ethyl‐2‐pyrrolidinyl)methyl]‐5‐(2[F‐18]fluoroethyl)‐2‐methoxybenzamide: A potential fluorine‐18 labeled PET radiotracer for dopamine D2 receptors
  Journal of Labelled Compounds and Radiopharmaceuticals, 1990
• Synthesis and in vitro affinity for dopamine D-2 receptor of N-fluorine-substituted analogs of eticlopride.
  CHEMICAL & PHARMACEUTICAL BULLETIN, 1989
• Determination of the novel quantitative structure-activity relationships descriptor .SIGMA.S.DEG. for di- and trisubstituted benzene derivatives.
  CHEMICAL & PHARMACEUTICAL BULLETIN, 1989
• Potential neuroleptic agents. 3. Chemistry and antidopaminergic properties of substituted 6-methoxysalicylamides
  Journal of Medicinal Chemistry, 1985
• Quantitative relationships between structure and pharmacokinetics of beta-adrenoceptor blocking agents in man
  Journal of Pharmacokinetics and Biopharmaceutics, 1984
• A New Substituent Constant, π, Derived from Partition Coefficients
  Journal of the American Chemical Society, 1964
• The Location of Electrostatic Charges in Kirkwood's Model of Organic Ions
  Journal of the American Chemical Society, 1957