‘Click chemistry’ synthesis of a library of 1,2,3-triazole-substituted galactose derivatives and their evaluation against Trypanosoma cruzi and its cell surface trans-sialidase
- 2 March 2010
- journal article
- research article
- Published by Elsevier in Bioorganic & Medicinal Chemistry
- Vol. 18 (7) , 2412-2427
- https://doi.org/10.1016/j.bmc.2010.02.053
Abstract
No abstract availableKeywords
This publication has 59 references indexed in Scilit:
- Nitric oxide donor trans‐[RuCl([15]aneN4)NO]2+ as a possible therapeutic approach for Chagas' diseaseBritish Journal of Pharmacology, 2010
- Novel ruthenium complexes as potential drugs for Chagas's disease: enzyme inhibition and in vitro/in vivo trypanocidal activityBritish Journal of Pharmacology, 2010
- Detailed insights from microarray and crystallographic studies into carbohydrate recognition by microneme protein 1 (MIC1) of Toxoplasma gondiiProtein Science, 2009
- Discovery of novel inhibitors of Trypanosoma cruzi trans-sialidase from in silico screeningBioorganic & Medicinal Chemistry Letters, 2009
- 2,3,4,6-Tetra-O-acetyl-α-D-glucopyranosyl azideActa Crystallographica Section C Crystal Structure Communications, 2008
- The war against influenza: discovery and development of sialidase inhibitorsNature Reviews Drug Discovery, 2007
- Glycosidase inhibition by 1-glycosyl-4-phenyl triazolesBioorganic & Medicinal Chemistry Letters, 2005
- A Potent and Highly Selective Inhibitor of Human α-1,3-Fucosyltransferase via Click ChemistryJournal of the American Chemical Society, 2003
- A Stepwise Huisgen Cycloaddition Process: Copper(I)-Catalyzed Regioselective “Ligation” of Azides and Terminal AlkynesAngewandte Chemie International Edition in English, 2002
- Hydrolase and sialyltransferase activities of Trypanosoma cruzi trans -sialidase towards NeuAc-α-2,3-Gal-β- O -PNPBioorganic & Medicinal Chemistry Letters, 2001