A bioisosteric approach to the discovery of indole carbinol androgen receptor ligands
- 1 November 2006
- journal article
- research article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 16 (21) , 5646-5649
- https://doi.org/10.1016/j.bmcl.2006.08.036
Abstract
No abstract availableKeywords
This publication has 11 references indexed in Scilit:
- Nonsteroidal tissue selective androgen receptor modulators: a promising class of clinical candidatesExpert Opinion on Therapeutic Patents, 2005
- Chemistry and Structural Biology of Androgen ReceptorChemical Reviews, 2005
- Discovery and Therapeutic Promise of Selective Androgen Receptor ModulatorsMolecular Interventions, 2005
- Bioisosterism: A Useful Strategy for Molecular Modification and Drug DesignCurrent Medicinal Chemistry, 2005
- Bioisosterism: Quantitation of Structure and Property EffectsChemistry & Biodiversity, 2004
- Biological function and mode of action of the androgen receptorPure and Applied Chemistry, 2003
- Molecular Biology of the Androgen ReceptorJournal of Clinical Oncology, 2002
- Bioisosterism: A Rational Approach in Drug DesignChemical Reviews, 1996
- An Efficient Synthesis of 1,2,9,9a-Tetrahydrocyclopropa[c]benz[e]indol-4-one CBI: An Enhanced and Simplified Analog of the CC-1065 and Duocarmycin Alkylation SubunitsThe Journal of Organic Chemistry, 1995
- Asymmetric hydroformylation of N-acyl 1-aminoacrylic acid derivatives by rhodium/chiral diphosphine catalystsTetrahedron: Asymmetry, 1991