Preparation of 14,15-secoestra-1,3,5(10)-trien-15-ynes, inhibitors of estradiol dehydrogenase
- 28 February 1989
- Vol. 53 (1-2) , 77-96
- https://doi.org/10.1016/0039-128x(89)90147-5
Abstract
No abstract availableKeywords
This publication has 30 references indexed in Scilit:
- Dehydrogenase inactivation by an enzyme-generated acetylenic ketone: identification of a lysyl enaminone by carbon-13 NMRJournal of the American Chemical Society, 1987
- Mechanism-based inactivation of 17.beta.,20.alpha.-hydroxysteroid dehydrogenase by an acetylenic secoestradiolBiochemistry, 1986
- Suicide Enzyme InactivatorsChemical & Engineering News, 1983
- Inactivation of Δ5-3-ketosteroid isomerase(s) from beef adrenal cortex by acetylenic ketosteroidsThe Journal of Steroid Biochemistry and Molecular Biology, 1982
- Suicide substrates: mechanism-based enzyme inactivatorsTetrahedron, 1982
- Inactivation of Δ5-3-oxo steroid isomerase with active-site-directed acetylenic steroidsBiochemical Journal, 1981
- Study of 3.alpha.,20.beta.-hydroxysteroid dehydrogenase with an enzyme-generated affinity alkylator: dual enzyme activity at a single active siteBiochemistry, 1980
- Synthesis of 14.beta.-fluoro steroidsThe Journal of Organic Chemistry, 1972
- Studies of Steroid Ring D Epoxides of Enol Acetates; A New Synthesis of Estriol and of Androstane-3β,16α,17β-triol1Journal of the American Chemical Society, 1954
- THE INTERCONVERSION OF ESTRONE AND ESTRADIOL BY HUMAN TISSUE SLICES1,2,3Endocrinology, 1953