Iron-catalysed Negishi coupling of benzylhalides and phosphates
- 11 December 2008
- journal article
- research article
- Published by Royal Society of Chemistry (RSC) in Chemical Communications
- No. 5,p. 600-602
- https://doi.org/10.1039/b818961g
Abstract
Iron-based catalysts containing either 1,2-bis(diphenylphosphino)benzene or 1,3-bis(diphenylphosphino)propane give excellent activity and good selectivity in the Negishi coupling of aryl zinc reagents with a range of benzylhalides and phosphates.Keywords
This publication has 35 references indexed in Scilit:
- Simple Palladium(II) Precatalyst for Suzuki−Miyaura Couplings: Efficient Reactions of Benzylic, Aryl, Heteroaryl, and Vinyl Coupling PartnersOrganic Letters, 2007
- Activation and functionalization of benzylic derivatives by palladium catalystsChemical Society Reviews, 2007
- Suzuki−Miyaura Cross-Coupling Reactions of Benzyl Halides with Potassium AryltrifluoroboratesThe Journal of Organic Chemistry, 2006
- Suzuki−Miyaura Cross-Coupling of Benzylic Phosphates with Arylboronic AcidsOrganic Letters, 2005
- Suzuki−Miyaura Cross-Coupling of Benzylic Carbonates with Arylboronic AcidsOrganic Letters, 2005
- Rational Design and Synthesis of Novel Dimeric Diketoacid-Containing Inhibitors of HIV-1 Integrase: Implication for Binding to Two Metal Ions on the Active Site of IntegraseJournal of Medicinal Chemistry, 2004
- Preliminary in vitro studies on two potent, water-soluble trimethoprim analogues with exceptional species selectivity against dihydrofolate reductase from Pneumocystis carinii and Mycobacterium aviumBioorganic & Medicinal Chemistry Letters, 2004
- The Structure and Synthesis of Tsitsikammafuran: A New Furanosesquiterpene from a South African Dysidea SpongeTetrahedron, 2000
- Conformationally Restricted Analogues of Trimethoprim: 2,6-Diamino-8-substituted Purines as Potential Dihydrofolate Reductase Inhibitors from Pneumocystis carinii and Toxoplasma gondiiJournal of Medicinal Chemistry, 1997
- Synthesis and Dihydrofolate Reductase Inhibitory Activities of 2,4-Diamino-5-deaza and 2,4-Diamino-5,10-dideaza Lipophilic AntifolatesJournal of Medicinal Chemistry, 1997