An SAR study for the non-peptide substance P receptor (NK1) antagonist, CP-96,345.
- 30 June 1992
- journal article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 2 (6) , 559-564
- https://doi.org/10.1016/s0960-894x(01)81197-5
Abstract
No abstract availableKeywords
This publication has 13 references indexed in Scilit:
- Tachykinin receptor types: Classification and membrane signalling mechanismsNeurochemistry International, 1991
- A Potent Nonpeptide Antagonist of the Substance P (NK 1 ) ReceptorScience, 1991
- Preparation and radiolabelling of CP-96,345, the first non-peptide substance P antagonistBioorganic & Medicinal Chemistry Letters, 1991
- Pharmacological analysis of [3H]‐senktide binding to NK3 tachykinin receptors in guinea‐pig ileum longitudinal muscle‐myenteric plexus and cerebral cortex membranesBritish Journal of Pharmacology, 1990
- The polyprotein nature of substance P precursorsBioEssays, 1989
- TachykininsAnnual Review of Neuroscience, 1988
- Multiple tachykinin binding sites in peripheral tissues and in brainEuropean Journal of Pharmacology, 1986
- Quinuclidine chemistry. 4. Diuretic properties of cis-3-amino-2-benzhydrylquinuclidineJournal of Medicinal Chemistry, 1975
- Quinuclidine chemistry. 2. Synthesis and antiinflammatory properties of 2-substituted benzhydryl-3-quinuclidinolsJournal of Medicinal Chemistry, 1974
- An unidentified depressor substance in certain tissue extractsThe Journal of Physiology, 1931