Whole cell catalysed kinetic resolution of 6-azabicyclo[3.2.0]hept-3-en-7-one: synthesis of (–)-cispentacin (FR 109615)
- 1 January 1991
- journal article
- research article
- Published by Royal Society of Chemistry (RSC) in Journal of the Chemical Society, Perkin Transactions 1
- No. 9,p. 2276-2277
- https://doi.org/10.1039/p19910002276
Abstract
Enantioselective hydrolysis of the β-lactam (±)-2 using Rhodococcus equi provided (1R,5S)-6azabicyclo[3.2.0] hept-3-en-7-one (+)-2, a precursor of the antifungal agent cispentacin.Keywords
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