Structural Analogues Of Aporphines Part 1: Synthesis of Apomorphines with the Catechol Moiety Replaced by 5‐membered Heterocycles
- 16 June 1982
- journal article
- research article
- Published by Wiley in Helvetica Chimica Acta
- Vol. 65 (4) , 1304-1309
- https://doi.org/10.1002/hlca.19820650421
Abstract
Analogues of apomorphine (1) having the catechol moiety replaced by pyrrole (→10, 18), pyrazole (→12), isoxazole (→13, 14), thiazole (→16) and thiadiazole (→20) ring systems have been synthesized from the key intermediate ketone 6.This publication has 8 references indexed in Scilit:
- Umsetzungen von Ketonen mit azavinylogen SäureamidenEuropean Journal of Inorganic Chemistry, 1975
- Chemische und pharmakologische Studien über Derivate des Benzo[de]chinolins (I). 8. Mitteilung über natürliche und synthetische IsochinolinderivateHelvetica Chimica Acta, 1973
- Lupinen‐Alkaloide, XXXIX. Addition von Butadiencarbonsäureester an cyclische ImineEuropean Journal of Inorganic Chemistry, 1967
- The Synthesis of 2,3,9,9a-Tetrahydro- 6-hydroxy-5-methoxy-1-methyl-1H-benzo- [d,e]quinolin-7(8H)-oneThe Journal of Organic Chemistry, 1964
- Über die anomale Reaktionsweise des 2‐Amino‐4.5‐trimethylen‐thiazolsEuropean Journal of Inorganic Chemistry, 1960
- Eine Synthese einfacher heterocyclischer VerbindungenEuropean Journal of Inorganic Chemistry, 1949
- THE CONSTITUTION OF THE NITRO-α-CARBOPYRROLIC ACIDS.2Journal of the American Chemical Society, 1915
- Eine neue und rationelle Indol‐Synthese. (Über das o‐Aldehydophenyl‐glycin. II)European Journal of Inorganic Chemistry, 1915