Resistance mutations at the lipid substrate binding site of Plasmodium falciparum protein farnesyltransferase
- 31 March 2007
- journal article
- Published by Elsevier in Molecular and Biochemical Parasitology
- Vol. 152 (1) , 66-71
- https://doi.org/10.1016/j.molbiopara.2006.11.012
Abstract
No abstract availableKeywords
This publication has 25 references indexed in Scilit:
- Thematic review series: Lipid Posttranslational Modifications. Fighting parasitic disease by blocking protein farnesylationJournal of Lipid Research, 2006
- Protein Farnesyltransferase Inhibitors Exhibit Potent Antimalarial ActivityJournal of Medicinal Chemistry, 2005
- The global distribution of clinical episodes of Plasmodium falciparum malariaNature, 2005
- Inhibitors of Farnesyltransferase: A Rational Approach to Cancer Chemotherapy?Journal of Medicinal Chemistry, 2004
- Farnesyltransferase inhibitorsSeminars in Oncology, 2004
- Design and Synthesis of Peptidomimetic Protein Farnesyltransferase Inhibitors as Anti-Trypanosoma brucei AgentsJournal of Medicinal Chemistry, 2003
- Protein Farnesyltransferase and Protein Prenylation inPlasmodium falciparumJournal of Biological Chemistry, 2002
- Yeast Protein Farnesyltransferase: A Pre-Steady-State Kinetic AnalysisBiochemistry, 1997
- Protein farnesyltransferase: kinetics of farnesyl pyrophosphate binding and product releaseBiochemistry, 1995
- Human Malaria Parasites in Continuous CultureScience, 1976